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| Return to: KESIMPTA (ofatumumab) | |
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| #Post#: 136-------------------------------------------------- | |
| Ofatumumab | |
| By: agate Date: January 25, 2014, 11:47 pm | |
| --------------------------------------------------------- | |
| Ofatumumab has reached only Phase 2 but here it is, a new drug | |
| that just might work. | |
| From PubMed, January 24, 2014: | |
| [quote]Neurology. 2014 Jan 22. | |
| Safety and efficacy of ofatumumab in relapsing-remitting | |
| multiple sclerosis: A phase 2 study | |
| Sorensen PS, Lisby S, Grove R, Derosier F, Shackelford S, | |
| Havrdova E, Drulovic J, Filippi M. | |
| Author information | |
| From the Danish Multiple Sclerosis Center (P.S.S.), | |
| Rigshospitalet, Copenhagen; Genmab (S.L.), Copenhagen, Denmark; | |
| GlaxoSmithKline (R.G.), Uxbridge, Middlesex, UK; GlaxoSmithKline | |
| (F.D.), Research Triangle Park; GlaxoSmithKline (S.S.), Raleigh, | |
| NC; Charles University (E.H.), Prague, Czech Republic; School of | |
| Medicine University of Belgrade (J.D.), Serbia; and San Raffaele | |
| Scientific Institute and Vita-Salute San Raffaele University | |
| (M.F.), Milan, Italy. | |
| OBJECTIVES: | |
| We present the first study to explore safety and efficacy of the | |
| human CD20 monoclonal antibody ofatumumab in relapsing-remitting | |
| multiple sclerosis (RRMS). | |
| METHODS: | |
| In this randomized, double-blind, placebo-controlled study, | |
| patients received 2 ofatumumab infusions (100 mg, 300 mg, or 700 | |
| mg) or placebo 2 weeks apart. At week 24, patients received | |
| alternate treatment. Safety and efficacy were assessed. | |
| RESULTS: | |
| Thirty-eight patients were randomized (ofatumumab/placebo, n = | |
| 26; placebo/ofatumumab, n = 12) and analyzed; 36 completed the | |
| study. Two patients in the 300-mg group withdrew from the study | |
| because of adverse events. No unexpected safety signals emerged. | |
| Infusion-related reactions were common on the first infusion day | |
| but not observed on the second infusion day. None of the | |
| patients developed human anti-human antibodies. Ofatumumab was | |
| associated with profound selective reduction of B cells as | |
| measured by CD19+ expression. New brain MRI lesion activity was | |
| suppressed (>99%) in the first 24 weeks after ofatumumab | |
| administration (all doses), with statistically significant | |
| reductions (p < 0.001) favoring ofatumumab found in new T1 | |
| gadolinium-enhancing lesions, total enhancing T1 lesions, and | |
| new and/or enlarging T2 lesions. | |
| CONCLUSIONS: | |
| Ofatumumab (up to 700 mg) given 2 weeks apart was not associated | |
| with any unexpected safety concerns and was well tolerated in | |
| patients with RRMS. MRI data suggest a clinically meaningful | |
| effect of ofatumumab for all doses studied. Results warrant | |
| further exploration of ofatumumab in RRMS. | |
| CLASSIFICATION OF EVIDENCE: | |
| This study provides Class II evidence that in patients with | |
| RRMS, ofatumumab compared with placebo does not increase the | |
| number of serious adverse events and decreases the number of new | |
| MRI lesions. | |
| PMID: 24453078[/quote] | |
| The abstract can be seen here | |
| http://www.ncbi.nlm.nih.gov/pubmed/24453078. | |
| #Post#: 916-------------------------------------------------- | |
| Novartis to buy ofatumumab from GlaxoSmithKline | |
| By: agate Date: August 28, 2015, 7:51 pm | |
| --------------------------------------------------------- | |
| From the New York Times, August 21, 2015: | |
| [quote]Novartis to Buy Multiple Sclerosis Drug From Glaxo | |
| By AMIE TSANG and ANDREW POLLACK | |
| Novartis bolstered its portfolio of multiple sclerosis | |
| treatments on Friday by agreeing to buy an experimental drug | |
| from GlaxoSmithKline for up to $1 billion, the company said. | |
| Novartis, the Swiss pharmaceutical giant, acquired the rights | |
| this year to use the drug, ofatumumab, to treat cancer, and | |
| sells it under the name Arzerra. This was part of a broader swap | |
| of assets completed in March, in which Novartis took over | |
| Glaxo�s cancer drugs and Glaxo took on much of Novartis�s | |
| vaccine business. | |
| The deal announced on Friday gives Novartis all remaining rights | |
| to ofatumumab, which is being developed to treat relapsing, | |
| remitting multiple sclerosis and other autoimmune conditions. | |
| Having the rights under one ownership would avoid the | |
| complications that could arise from having two companies selling | |
| the same drug for different uses. The deal also bolsters a | |
| portfolio of drugs Novartis is developing for multiple | |
| sclerosis, centered around its blockbuster pill Gilenya. | |
| Novartis will pay $300 million upfront to Glaxo and another $200 | |
| million once late-stage clinical trials start. Novartis would | |
| make payments of up to $534 million on top of that, depending on | |
| whether development targets are reached. The company will also | |
| pay royalties of up to 12 percent to Glaxo on any future net | |
| sales of the drug. | |
| �Novartis is pleased to further reinforce our commitment to | |
| neuroscience and to add an exciting new treatment to our strong | |
| MS portfolio,� David Epstein, the division head of Novartis | |
| Pharmaceuticals, said in a news release. | |
| In addition to Gilenya, Novartis sells a multiple sclerosis drug | |
| called Extavia and recently began marketing a generic version of | |
| Teva�s Copaxone, one of the most widely used drugs for the | |
| disease. It also has some other drugs in development. Gilenya | |
| could lose patent protection starting in 2019. So filling the | |
| loss could be another reason for Novartis to want a new drug. | |
| But the market for multiple sclerosis drugs is crowded, which | |
| could limit the sales any new drug like ofatumumab could have. | |
| Moreover, ofatumumab is only now ready to enter late-stage | |
| clinical trials, putting it a couple of years behind | |
| ocrelizumab, a similar drug being developed by Roche. | |
| Both drugs deplete B cells, which are white blood cells that are | |
| part of the immune system. B cells are necessary to fight | |
| infections, but if they go awry, they can contribute to | |
| autoimmune diseases like multiple sclerosis or to lymphomas. | |
| Both drugs bind to the same molecule on the surface of B cells � | |
| known as CD20 � as Roche�s big-selling cancer drug Rituxan. | |
| Rituxan is not approved for multiple sclerosis, but it is | |
| approved to treat rheumatoid arthritis, another autoimmune | |
| disease. | |
| Ofatumumab, a type of protein called a monoclonal antibody, was | |
| developed initially by Genmab, a Danish biotechnology company, | |
| which receives royalties on sales. | |
| David Redfern, the chief strategy officer at Glaxo, said in a | |
| news release that the sale would allow the company to focus on | |
| core areas, including H.I.V., oncology and vaccines. | |
| �We are pleased to have completed this transaction to divest the | |
| remaining rights in ofatumumab, crystallizing significant | |
| additional value for G.S.K. shareholders,� Mr. Redfern said. | |
| The deal is expected to be completed by the end of the | |
| year.[/quote] | |
| #Post#: 2064-------------------------------------------------- | |
| Re: (Abst.) Subcutaneous ofatumumab in patients w/RRMS: The MIRR | |
| OR study | |
| By: agate Date: April 27, 2018, 7:28 pm | |
| --------------------------------------------------------- | |
| From PubMed, April 27, 2018--"Subcutaneous ofatumumab in | |
| patients with RRMS: The MIRROR study": | |
| https://www.ncbi.nlm.nih.gov/pubmed/29695594 | |
| #Post#: 2635-------------------------------------------------- | |
| Market share drama with ofatumumab a new player | |
| By: agate Date: August 30, 2019, 10:03 am | |
| --------------------------------------------------------- | |
| A couple of drug companies are competing with each other. It's | |
| Ocrevus against ofatumumab according to this press release from | |
| Reuters (August 29, 2019)--"Novartis Takes Aim at Roche's Star | |
| MS Drug": | |
| https://reut.rs/2ZttMEj | |
| #Post#: 2652-------------------------------------------------- | |
| (ECTRIMS) Ofatumumab may be competing with ocrelizumab | |
| By: agate Date: September 16, 2019, 5:22 pm | |
| --------------------------------------------------------- | |
| From Medscape (September 16, 2019)--"Ofatumumab impresses in MS: | |
| Competition with ocrelizumab soon?" | |
| https://www.medscape.com/viewarticle/918478#vp_1 | |
| #Post#: 2788-------------------------------------------------- | |
| Update on ofatumumab (OMB157) | |
| By: agate Date: January 22, 2020, 1:32 am | |
| --------------------------------------------------------- | |
| An update on ofatumumab--from Nasdaq.com (January 21, 2020), | |
| "Novartis gets approval for MS drug Mayzent in Europe." (The | |
| article contains information about ofatumumab.) | |
| https://www.nasdaq.com/articles/novartis-nvs-gets-approval-for-ms-drug-mayzent-… | |
| #Post#: 2831-------------------------------------------------- | |
| (ACTRIMS) Ofatumumab self-injector pen results equivalent to inf | |
| usion... | |
| By: agate Date: March 2, 2020, 11:57 pm | |
| --------------------------------------------------------- | |
| From Multiple Sclerosis News Today, a report from the annual | |
| ACTRIMS conference held February 27-29, 2020, "Ofatumumab | |
| self-injector pen results equivalent to infusion, trial shows": | |
| http://bit.ly/39uyXFq | |
| #Post#: 2988-------------------------------------------------- | |
| (NEJM abstract) Ofatumumab shows better results than Aubagio | |
| By: agate Date: August 6, 2020, 10:01 am | |
| --------------------------------------------------------- | |
| From the New England Journal of Medicine (August 6, | |
| 2020)--"Ofatumumab versus Teriflunomide in Multiple Sclerosis": | |
| https://www.nejm.org/doi/full/10.1056/NEJMoa1917246?query=TOC | |
| It might be worth noting that the study was funded by Novartis. | |
| #Post#: 3001-------------------------------------------------- | |
| FDA approval of Kesimpta (ofatumumab) | |
| By: agate Date: August 21, 2020, 11:48 am | |
| --------------------------------------------------------- | |
| Another MS drug to add to the collection of FDA-approved MS | |
| treatments--a press release from Novartis, dated August 20, | |
| 2020: | |
| https://bit.ly/2QfChfG | |
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